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Can Subutex Really Block Opiates? How Long?

When this question is asked, it helps to bear in mind that the long-term use of opiates is almost guaranteed to alter the functions of the brain in countless ways. Generally, the medications used to block opiates can aid in meeting a few of the challenges that drug addicts face in the time of recovery, although not all of them.

It should be known that the effects of opiates especially in long-term addictions can persist even long after the user stops taking medications. Moreover, if the user avoids any form of treatment, the individual would find it extremely difficult in the long run to abstain from the drug on a progressive basis.

One of the various FDA approved medications used for the treatment of opiate addiction, the Subutex presents established therapeutic effects that some drugs like methadone cannot execute. Subutex, unlike methadone, creates a two-fold effect in how the drug interacts with the opioid receptors in the human brain.

The After-Effect Of Opiate Addiction

The human body actually has its own opioid system for regulating sensations of pleasure and pain on a continuous basis. The opioid system also digs deeper into the learning and rewards system of the brain. Therefore, opiate addiction can leave these bodily functions in a state of disarray.

Opiates activate the opioid receptor sites found in the many cells of the brain, the central nervous system, and the gastrointestinal tract. When a person ingests opiates, the drugs tend to interfere with the body’s own system of pain management, completely redefining how the brain should interpret reward and pleasure.

Years of opiate abuse can lead the normal functions of the brain and central nervous system to partially if not fully rely on opiates for regular bodily functions. If a user decides to cease the medication use or abuse, professional treatment is essentially required.

Subutex & Mechanism Of Action

The question ‘How long does Subutex block opiates?’ can best be confronted with the drug’s effectiveness in assisting recovery. The withdrawal effects and cravings for opiates are two of the biggest obstacles faced during long-term abstinence and this is what Subutex aims to address.

  • The Substance Abuse and Mental Health Services Administration reveals that Subutex is usually found in the brand name buprenorphine, which is the newest treatment drug for opiate addiction in the market.
  • Subutex can actually interact with the very same cells that opiates interacted with, only in the opposite way.
  • The drug functions mostly like methadone in the therapeutic benefits that it gives.
  • Both Subutex and methadone drugs can support cell functions and also restore the normal endorphin levels in the body. During treatment, addicted individuals can gain a form of relief from their withdrawal symptoms and after-effects of drug cravings.

Subutex acts as an opioid partial antagonist, which means that it can both activate the cell site receptors and block the affected ones. On the other hand, methadone is a full agonist, unable to block opiates at all. Subutex creates a strong bond with the cell receptors. Once Subutex goes into a cell receptor, opiates like morphine and heroin will no longer be able to activate these sites.

The “ceiling effect” of the drug is what can diminish the possibility of abuse and addiction. The Subutex’s ability to activate the cell site receptors can max out after a certain dose level. Hence, it will be difficult to get “high” in the event that a relapse occurs.

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